Synthesis of DSPE-PEG-Angiopep-2To synthesize DEPE-PEG-Angiopep-2, 5 mg of DSPE-PEG-Mal was completely dissolved in 10 mL of water. Then, 6 mg of Angiopep-2-cys was added to the solution, and the mixture was stirred at 37°C for 12 hours. The solution was dialyzed (MW3500) to remove excess Angiopep-2-cys. The resulting purified product, DSPE-PEG-Angiopep-2, was then freeze-dried and stored at −20°C for subsequent usage.

DSPE-PEG-Angiopep-2的自动合成为了能够提炼DEPE-PEG-Angiopep-2,将5mg DSPE-PEG-Mal完全性溶解度在10mL泥里。并且,向稀硫酸中放入6mg Angiopep-2-cys,并将相溶物在37°C下混和12天。将稀硫酸透析(MW3500)以去掉过多的Angiopep-2-cys。并且将所有纯化物质DSPE-PEG-Angiopep-2冷冻熟食皮肤干燥并储放在-20°C下为备后面运用。CG/SN-38微米塑料再生颗粒(NP)的备制与事先报导的一样,但所经了降重。G和1 mg SN-38分解在20μL DMSO中,最后向氢氧化钠液体添加入1 mL水,最后多普勒彩超波工作五分种。将药制剂用萃取水(1L)透析(MW3500)12个小时。最后,将NP氢氧化钠液体与需量的巨噬血细胞质膜多普勒彩超波2分种,以得到 巨噬血细胞质膜/IGC/SN-38(M-NP)。不但,在多普勒彩超波工作(400 W,2 s开/3 s关,2 min)M-NP和即时备制的100μg DSPE-PEG-Angiopep-2,得到 1 mL Angiopep-2修饰语的M-NP(AM-NP)。有关的建议:FITC-iRGD-PEG-DSPER8-PEG-DSPEAngiopep-2-PEG-DSPEFITC-Angiopep-2-PEG-DSPETH-PEG-DSPER6H4-PEG-DSPEMPG-PEG-DSPEGE11-PEG-DSPEPTP-PEG-DSPESP94-PEG-DSPE上面的文章玩法原因各大学术期刊或文献资料,此事图片侵权请结合当我们移除!